SCHEMBL28934545

SCHEMBL28934545

N#Cc1ccc(-c2nnc(N[C@@H]3CCCN(S(=O)(=O)C4CC4)C3)c3ccccc23)c(O)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 11/20 0.49
IRAK4 Q9NWZ3 1/20 0.41
ALDH1A1 P00352 2/20 0.40
IL1B P01584 1/20 0.39
CYP11B1 P15538 3/20 0.38
CYP11B2 P19099 3/20 0.38
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 1/20 0.37
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28934549 1.00 NLRP3 (0.49) NLRP3IRAK4ALDH1A1IL1BCYP11B1
SCHEMBL25864163 0.91 NLRP3 (0.45) NLRP3ALDH1A1IL1BCYP11B1CYP11B2
SCHEMBL28934539 0.91 NLRP3 (0.51) NLRP3IRAK4ALDH1A1IL1BJAK2
SCHEMBL30108776 0.91 NLRP3 (0.51) NLRP3IRAK4ALDH1A1IL1BJAK2
SCHEMBL28934535 0.91 NLRP3 (0.51) NLRP3IRAK4ALDH1A1IL1BJAK2
SCHEMBL30108648 0.85 NLRP3 (0.62) NLRP3IL1B
SCHEMBL28934482 0.85 NLRP3 (0.62) NLRP3IL1B
SCHEMBL28934477 0.85 NLRP3 (0.62) NLRP3IL1B
SCHEMBL28934737 0.84 NLRP3 (0.50) NLRP3IRAK4IL1BKDM4EHSD17B10
SCHEMBL28934734 0.84 NLRP3 (0.50) NLRP3IRAK4IL1BKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed