SCHEMBL25866149

SCHEMBL25866149

O=c1oc2ccc(Br)cc2n1C1COC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBX7 O95931 1/20 0.38
CDYL2 Q8N8U2 1/20 0.38
CDYL Q9Y232 1/20 0.38
CDY1; CDY1B Q9Y6F8 1/20 0.38
CHRM4 P08173 7/20 0.37
CHRM5 P08912 7/20 0.37
CHRM1 P11229 7/20 0.37
CHRM3 P20309 7/20 0.37
CHRM2 P08172 6/20 0.37
SIGMAR1 Q99720 1/20 0.37
NPC1 O15118 1/20 0.37
PIM1 P11309 1/20 0.36
ASAH1 Q13510 1/20 0.36
HPGD P15428 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25310581 0.85 NPC1 (0.40) CBX7CDYL2CDYLCDY1; CDY1BCHRM4
SCHEMBL25867651 0.82 SIGMAR1 (0.40) CBX7CDYL2CDYLCDY1; CDY1BCHRM4
SCHEMBL20117054 0.82 CHRM2 (0.53) CHRM4CHRM5CHRM1CHRM3CHRM2
SCHEMBL30476259 0.73 USP30 (0.44) ALDH1A1
SCHEMBL30988527 0.72 OPRM1 (0.56) CHRM4CHRM5CHRM1CHRM3CHRM2
SCHEMBL31426196 0.72 CRBN (0.54) CHRM2ALDH1A1TSHR
SCHEMBL31426197 0.72 CRBN (0.54) CHRM2ALDH1A1TSHR
SCHEMBL614398 0.70 SIGMAR1 (0.47) CBX7CDYL2CDYLCDY1; CDY1BSIGMAR1
SCHEMBL5546317 0.70 SIGMAR1 (0.44) CBX7CDYL2CDYLCDY1; CDY1BSIGMAR1
SCHEMBL29704410 0.70 SIGMAR1 (0.47) CBX7CDYL2CDYLCDY1; CDY1BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134656-A1 PEPTIDYL NITRILE COMPOUND AND USE THEREOF 上海壹典医药科技开发有限公司 2023-07-20 WO disclosed
CN-116332937-A Dipeptidyl peptidase I inhibitors and uses thereof 杭州邦顺制药有限公司 2023-06-27 CN disclosed