SCHEMBL25867651

SCHEMBL25867651

CN1CC(n2c(=O)oc3ccc(Br)cc32)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.40
CHRM4 P08173 6/20 0.38
CHRM5 P08912 6/20 0.38
CHRM1 P11229 6/20 0.38
CHRM3 P20309 6/20 0.38
CHRM2 P08172 5/20 0.38
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
CBX7 O95931 1/20 0.37
CDYL2 Q8N8U2 1/20 0.37
CDYL Q9Y232 1/20 0.37
CDY1; CDY1B Q9Y6F8 1/20 0.37
PIK3CD O00329 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 2/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
ASAH1 Q13510 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25866149 0.82 CBX7 (0.38) SIGMAR1CHRM4CHRM5CHRM1CHRM3
SCHEMBL25310581 0.82 NPC1 (0.40) SIGMAR1CHRM4CHRM5CHRM1CHRM3
SCHEMBL30476259 0.78 USP30 (0.44)
SCHEMBL29704410 0.75 SIGMAR1 (0.47) SIGMAR1CBX7CDYL2CDYLCDY1; CDY1B
SCHEMBL614398 0.75 SIGMAR1 (0.47) SIGMAR1CBX7CDYL2CDYLCDY1; CDY1B
SCHEMBL25309770 0.74 L3MBTL1 (0.37) SIGMAR1CHRM4CHRM5CHRM1CHRM3
SCHEMBL31426197 0.69 CRBN (0.54) CHRM2DDB1CRBN
SCHEMBL31426196 0.69 CRBN (0.54) CHRM2DDB1CRBN
SCHEMBL782891 0.69 SIGMAR1 (0.57) SIGMAR1CBX7CDYL2CDYLCDY1; CDY1B
SCHEMBL5546317 0.68 SIGMAR1 (0.44) SIGMAR1CBX7CDYL2CDYLCDY1; CDY1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134656-A1 PEPTIDYL NITRILE COMPOUND AND USE THEREOF 上海壹典医药科技开发有限公司 2023-07-20 WO disclosed