SCHEMBL2586615

SCHEMBL2586615

NC(=O)n1c(Cc2ccccc2)c(P(=S)(c2ccccc2)c2ccccc2)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 9/20 0.54
REN P00797 1/20 0.41
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HTR7 P34969 4/20 0.35
PLA2G10 O15496 1/20 0.35
PLA2G2A P14555 1/20 0.35
AGTR1 P30556 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590909 0.70 NPSR1 (1.00) NPSR1KDM4EALDH1A1
SCHEMBL31210085 0.66 POLB (0.61) NPSR1KDM4EALDH1A1HPGD
SCHEMBL10879830 0.66 POLB (0.61) NPSR1KDM4EALDH1A1HPGD
SCHEMBL28460971 0.66 KDM4E (0.46) RENKDM4EALDH1A1HPGDHTR7
SCHEMBL2595693 0.64 NPSR1 (1.00) NPSR1KDM4EALDH1A1HPGD
SCHEMBL2587268 0.63 NPSR1 (0.63) NPSR1KDM4EALDH1A1PLA2G2A
SCHEMBL2593998 0.63 NPSR1 (0.63) NPSR1ALDH1A1
SCHEMBL31590097 0.62 P2RX4 (0.56) NPSR1KDM4EALDH1A1HPGD
SCHEMBL2586743 0.60 NPSR1 (0.58) NPSR1KDM4EALDH1A1PLA2G2A
Diphenylmethane SCHEMBL8743340 0.60 PLA2G10 (0.71) PLA2G10PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137220-A1 SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-11-03 WO disclosed