SCHEMBL25866228

SCHEMBL25866228

Brc1ccc2c(c1)C1(CNC1)OC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 2/20 0.37
ASIC3 Q9UHC3 1/20 0.37
CMA1 P23946 1/20 0.36
AHR P35869 1/20 0.36
TDP2 O95551 1/20 0.34
BACE1 P56817 1/20 0.34
KDM1A O60341 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
CHEK2 O96017 1/20 0.33
ROS1 P08922 1/20 0.33
MARK3 P27448 1/20 0.33
LTK P29376 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
MINK1 Q8N4C8 1/20 0.33
AURKB Q96GD4 1/20 0.33
PBK Q96KB5 1/20 0.33
STK17A Q9UEE5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30098011 0.88 PNMT (0.40) PNMTASIC3CMA1AHRTDP2
SCHEMBL15505712 0.88 PNMT (0.40) PNMTASIC3CMA1AHRTDP2
Hydrochloric Acid SCHEMBL19616590 0.86 PNMT (0.39) PNMTASIC3CMA1AHRTDP2
SCHEMBL31515349 0.83 KDM1A (0.40) CMA1AHRTDP2KDM1A
SCHEMBL18373201 0.83 HTR2C (0.40) PNMTASIC3CMA1AHRTDP2
SCHEMBL30954699 0.80 KDM1A (0.38) CMA1AHRBACE1KDM1A
SCHEMBL25866296 0.80 BACE1 (0.37) CMA1AHRTDP2BACE1KDM1A
SCHEMBL30954718 0.77 LMNA (0.41) CMA1AHRBACE1KDM1A
SCHEMBL25866229 0.76 BRD4 (0.34) BACE1KDM1A
SCHEMBL30954707 0.76 BACE1 (0.39) CMA1AHRBACE1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024125488-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF 浙江海正药业股份有限公司 2024-06-20 WO disclosed
WO-2023134656-A1 PEPTIDYL NITRILE COMPOUND AND USE THEREOF 上海壹典医药科技开发有限公司 2023-07-20 WO disclosed