SCHEMBL2586836

SCHEMBL2586836

O=CCc1cccc2cccc-2c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGXT P21549 2/20 0.45
PTGS2 P35354 2/20 0.45
PRKCI P41743 1/20 0.44
BCL2 P10415 1/20 0.43
AOC3 Q16853 3/20 0.41
GGPS1 O95749 2/20 0.41
MMP3 P08254 1/20 0.40
GPR84 Q9NQS5 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
GPR52 Q9Y2T5 1/20 0.38
NR4A2 P43354 1/20 0.38
ACMSD Q8TDX5 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
CHKA P35790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1420024 0.96 AGXT (0.52) AGXTPTGS2PRKCIBCL2AOC3
SCHEMBL13186526 0.88 TAAR1 (0.48) AGXTPTGS2BCL2AOC3GGPS1
SCHEMBL1513827 0.86 HSD17B1 (0.54) MMP3GPR84
SCHEMBL5148894 0.85 CHKA (0.40) AGXTPTGS2PRKCIBCL2AOC3
SCHEMBL12345478 0.85 MAOB (0.39)
SCHEMBL6276471 0.84 CHKA (0.53) PTGS2AOC3CHKA
SCHEMBL4060950 0.81 CLK4 (0.46)
SCHEMBL3604987 0.81 PRMT6 (0.59) PRMT6ACMSD
SCHEMBL21368935 0.81 MAOB (0.51) AGXT
SCHEMBL16398826 0.81 MAOB (0.50) AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571879-A1 HETEROBIARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F.HOFFMANN-LA ROCHE AG (CH) 2013-03-27 EP disclosed
WO-2011134877-A1 HETEROBIARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-03 WO disclosed