SCHEMBL25877728

SCHEMBL25877728

COc1ccc(C)c(-c2ccnc(N)c2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.64
GSK3B P49841 1/20 0.59
NOS3 P29474 2/20 0.59
NOS1 P29475 2/20 0.59
NOS2 P35228 2/20 0.59
CDC7 O00311 1/20 0.47
PIM1 P11309 1/20 0.46
CDK9 P50750 1/20 0.46
DYRK2 Q92630 1/20 0.46
DYRK1B Q9Y463 1/20 0.46
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
TLR8 Q9NR97 1/20 0.43
ABL1 P00519 3/20 0.43
ROCK2 O75116 3/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25877903 0.84 DYRK1A (0.49) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL22272613 0.81 DYRK1A (0.46) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL22272939 0.80 DYRK1A (0.44) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL22272941 0.80 MAOA (0.45) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL30091626 0.80 DYRK1A (0.44) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL23927511 0.79 TSHR (0.46) DYRK1AGSK3BKDM4ECYP3A4CYP2D6
SCHEMBL25877820 0.79 DYRK1A (0.43) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL30091686 0.79 TSHR (0.46) DYRK1AGSK3BKDM4ECYP3A4CYP2D6
SCHEMBL22272533 0.78 DYRK1A (0.43) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL17054241 0.78 CYP11B2 (0.55) CYP11B1CYP11B2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138433-A2 AMIDE COMPOUND HAVING RIPK1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR, AND USE THEREOF 中国科学院上海药物研究所 2023-07-27 WO disclosed