SCHEMBL25879884

SCHEMBL25879884

CNC(=O)c1cc(Nc2ncc3ccc(C#N)cc3n2)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.39
CCNA2 P20248 2/20 0.39
CDK2 P24941 2/20 0.39
CDK7 P50613 2/20 0.39
CCNH P51946 2/20 0.39
MNAT1 P51948 2/20 0.39
CCNK O75909 1/20 0.39
CDK12 Q9NYV4 1/20 0.39
MAP4K1 Q92918 1/20 0.39
BRAF P15056 5/20 0.37
MAP3K5 Q99683 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
PTK2 Q05397 1/20 0.36
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CREBBP Q92793 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25879705 0.92 BRAF (0.43) SCN9ABRAFMAP3K5
SCHEMBL30512135 0.92 BRAF (0.43) SCN9ABRAFMAP3K5
SCHEMBL25881879 0.85 CDK7 (0.42) SCN9ACCNA2CDK2CDK7CCNH
SCHEMBL30512101 0.85 CDK7 (0.42) SCN9ACCNA2CDK2CDK7CCNH
SCHEMBL25881870 0.85 ALDH1A1 (0.41) CDK2BRAFMAP3K5CCNCCDK8
SCHEMBL25881895 0.84 CREBBP (0.46) BRAFMAP3K5CCNCCDK8PTK2
SCHEMBL25879550 0.82 MAP3K5 (0.54) CDK2BRAFMAP3K5CCNCCDK8
SCHEMBL30512112 0.82 MAP3K5 (0.54) CDK2BRAFMAP3K5CCNCCDK8
SCHEMBL25882093 0.82 BRAF (0.37) CDK2MAP4K1BRAFMAP3K5CCNC
SCHEMBL25881893 0.82 BRAF (0.37) CDK2BRAFMAP3K5CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed