SCHEMBL25879550

SCHEMBL25879550

CNC(=O)c1cc(Nc2ncc3ccccc3n2)c[nH]1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 2/20 0.54
BRAF P15056 12/20 0.47
ROCK1 Q13464 1/20 0.42
AURKA O14965 2/20 0.41
CDK2 P24941 2/20 0.41
MAPK1 P28482 1/20 0.41
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
KMT2A Q03164 1/20 0.40
SYK P43405 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30512112 1.00 MAP3K5 (0.54) MAP3K5BRAFROCK1AURKACDK2
SCHEMBL25880239 0.87 CCNC (0.48) MAP3K5BRAFCCNCCDK8
SCHEMBL25881961 0.86 MAP3K5 (0.54) MAP3K5BRAFROCK1AURKACDK2
SCHEMBL30512136 0.86 MAP3K5 (0.54) MAP3K5BRAFROCK1AURKACDK2
SCHEMBL25879561 0.86 BRAF (0.45) MAP3K5BRAFAURKACDK2CCNC
SCHEMBL25880438 0.86 CCNC (0.41) MAP3K5BRAFCCNCCDK8SYK
SCHEMBL30512101 0.86 CDK7 (0.42) MAP3K5BRAFCDK2CCNCCDK8
SCHEMBL25881879 0.86 CDK7 (0.42) MAP3K5BRAFCDK2CCNCCDK8
SCHEMBL25881870 0.86 ALDH1A1 (0.41) MAP3K5BRAFAURKACDK2MAPK1
SCHEMBL25881661 0.86 MAP3K5 (0.48) MAP3K5BRAFROCK1CDK2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed