SCHEMBL25880438

SCHEMBL25880438

CNC(=O)c1cc(Nc2ncc3ncccc3n2)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
PLK1 P53350 1/20 0.41
BRAF P15056 8/20 0.41
SYK P43405 6/20 0.41
MAP3K5 Q99683 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
NUDT1 P36639 1/20 0.38
CREBBP Q92793 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30512112 0.86 MAP3K5 (0.54) CCNCCDK8BRAFSYKMAP3K5
SCHEMBL25879550 0.86 MAP3K5 (0.54) CCNCCDK8BRAFSYKMAP3K5
SCHEMBL25880440 0.84 CCNC (0.41) CCNCCDK8PLK1BRAFSYK
SCHEMBL25880239 0.83 CCNC (0.48) CCNCCDK8BRAFMAP3K5CREBBP
SCHEMBL30512101 0.80 CDK7 (0.42) CCNCCDK8PLK1BRAFSYK
SCHEMBL25881870 0.80 ALDH1A1 (0.41) CCNCCDK8BRAFMAP3K5CREBBP
SCHEMBL25879561 0.80 BRAF (0.45) CCNCCDK8BRAFMAP3K5
SCHEMBL25881879 0.80 CDK7 (0.42) CCNCCDK8PLK1BRAFSYK
SCHEMBL25881895 0.79 CREBBP (0.46) CCNCCDK8BRAFMAP3K5CREBBP
SCHEMBL25879708 0.79 BRAF (0.52) BRAFMAP3K5CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed