SCHEMBL2588928

SCHEMBL2588928

Clc1cccc(Nc2nc(NCc3cccc(Br)c3)c3ccccc3n2)c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 2/20 0.65
APP P05067 4/20 0.60
PDE5A O76074 3/20 0.58
RAD52 P43351 1/20 0.53
MAPT P10636 2/20 0.52
KMT2A Q03164 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
PKM P14618 1/20 0.52
UBE2N P61088 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
RCE1 Q9Y256 1/20 0.52
SLC2A1 P11166 1/20 0.52
MEN1 O00255 1/20 0.50
GAA P10253 1/20 0.50
CTNNB1 P35222 1/20 0.49
TCF7L2 Q9NQB0 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2592287 0.92 SOS1 (0.71) SOS1APPPDE5ARAD52MAPT
SCHEMBL2583209 0.91 SOS1 (0.72) SOS1APPPDE5ARAD52MAPT
SCHEMBL2587225 0.90 SOS1 (0.66) SOS1APPPDE5ARAD52MAPT
SCHEMBL2588903 0.89 SOS1 (0.72) SOS1APPPDE5ARAD52MAPT
SCHEMBL2584997 0.87 SOS1 (0.65) SOS1APPPDE5ARAD52MAPT
SCHEMBL2587460 0.87 SOS1 (0.65) SOS1APPPDE5ARAD52MAPT
SCHEMBL2588890 0.87 SOS1 (0.70) SOS1APPPDE5ARAD52MAPT
SCHEMBL2590464 0.85 SLC2A1 (0.66) SOS1APPPDE5AMAPTKMT2A
SCHEMBL12176225 0.84 RAD52 (0.68) SOS1APPPDE5ARAD52MAPT
SCHEMBL2587416 0.84 RAD52 (0.76) APPRAD52MAPTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed