SCHEMBL2587460

SCHEMBL2587460

Cc1cccc(CNc2nc(Nc3cccc(Cl)c3)nc3ccccc23)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 2/20 0.65
LMNA P02545 6/20 0.61
MAPT P10636 6/20 0.61
MAPK1 P28482 6/20 0.61
ALDH1A1 P00352 4/20 0.61
KMT2A Q03164 4/20 0.61
USP2 O75604 3/20 0.61
HPGD P15428 2/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
NPSR1 Q6W5P4 2/20 0.61
NR2F2 P24468 1/20 0.61
APP P05067 3/20 0.60
PDE5A O76074 2/20 0.58
KDM4E B2RXH2 4/20 0.55
CYP1A2 P05177 4/20 0.55
CYP3A4 P08684 4/20 0.55
TSHR P16473 4/20 0.55
CYP2C19 P33261 4/20 0.55
HIF1A Q16665 3/20 0.55
MEN1 O00255 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2592287 0.92 SOS1 (0.71) SOS1LMNAMAPTALDH1A1KMT2A
SCHEMBL2583209 0.91 SOS1 (0.72) SOS1LMNAMAPTMAPK1ALDH1A1
SCHEMBL2588902 0.90 SOS1 (0.66) SOS1LMNAMAPTMAPK1ALDH1A1
SCHEMBL12176293 0.89 SOS1 (0.72) SOS1LMNAMAPTMAPK1ALDH1A1
SCHEMBL2584997 0.87 SOS1 (0.65) SOS1LMNAMAPTALDH1A1KMT2A
SCHEMBL2588928 0.87 SOS1 (0.65) SOS1LMNAMAPTALDH1A1KMT2A
SCHEMBL2588890 0.87 SOS1 (0.70) SOS1LMNAMAPTALDH1A1KMT2A
SCHEMBL2590464 0.87 SLC2A1 (0.66) SOS1LMNAMAPTMAPK1ALDH1A1
SCHEMBL12175983 0.84 RAD52 (0.76) LMNAMAPTMAPK1ALDH1A1KMT2A
SCHEMBL2587390 0.84 SOS1 (0.66) SOS1LMNAMAPTMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed