SCHEMBL2590464

SCHEMBL2590464

COc1cccc(CNc2nc(Nc3cccc(Cl)c3)nc3ccccc23)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.66
KDM4E B2RXH2 2/20 0.63
HTT P42858 2/20 0.63
TAAR1 Q96RJ0 1/20 0.63
APP P05067 2/20 0.62
SOS1 Q07889 1/20 0.62
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
MAPT P10636 2/20 0.57
MAPK1 P28482 2/20 0.56
ALDH1A1 P00352 2/20 0.56
USP2 O75604 1/20 0.56
LMNA P02545 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
TSHR P16473 1/20 0.56
CYP2C19 P33261 1/20 0.56
HSD17B10 Q99714 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590586 0.91 SLC2A1 (0.73) SLC2A1KDM4EHTTTAAR1APP
SCHEMBL2592287 0.90 SOS1 (0.71) SLC2A1KDM4EAPPSOS1MEN1
SCHEMBL2583209 0.88 SOS1 (0.72) SLC2A1KDM4EHTTAPPSOS1
SCHEMBL2587460 0.87 SOS1 (0.65) SLC2A1KDM4EAPPSOS1MEN1
SCHEMBL2587104 0.85 APP (0.76) SLC2A1KDM4EAPPMEN1KMT2A
SCHEMBL2588928 0.85 SOS1 (0.65) SLC2A1KDM4EAPPSOS1MEN1
SCHEMBL2584997 0.85 SOS1 (0.65) SLC2A1KDM4EAPPSOS1KMT2A
SCHEMBL2588890 0.84 SOS1 (0.70) SLC2A1KDM4EAPPSOS1KMT2A
SCHEMBL2588902 0.83 SOS1 (0.66) SLC2A1KDM4EHTTAPPSOS1
SCHEMBL2587500 0.83 SLC2A1 (0.65) SLC2A1KDM4EHTTTAAR1SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed