SCHEMBL2587225

SCHEMBL2587225

Clc1cccc(Nc2nc(NCc3ccc(Br)cc3)c3ccccc3n2)c1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 2/20 0.66
PDE5A O76074 2/20 0.59
EGFR P00533 1/20 0.56
APP P05067 3/20 0.56
CTNNB1 P35222 1/20 0.55
TCF7L2 Q9NQB0 1/20 0.55
RAD52 P43351 1/20 0.54
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
KMT2A Q03164 2/20 0.54
HTT P42858 1/20 0.54
NTRK1 P04629 1/20 0.53
LMNA P02545 1/20 0.53
PKM P14618 1/20 0.53
UBE2N P61088 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RCE1 Q9Y256 1/20 0.53
SLC2A1 P11166 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2588890 0.92 SOS1 (0.70) SOS1PDE5AAPPCTNNB1TCF7L2
SCHEMBL2583209 0.92 SOS1 (0.72) SOS1PDE5AAPPCTNNB1TCF7L2
SCHEMBL2588928 0.90 SOS1 (0.65) SOS1PDE5AAPPCTNNB1TCF7L2
SCHEMBL2588902 0.89 SOS1 (0.66) SOS1PDE5AAPPCTNNB1TCF7L2
SCHEMBL2590218 0.89 SOS1 (0.66) SOS1PDE5AAPPCTNNB1TCF7L2
SCHEMBL2592287 0.89 SOS1 (0.71) SOS1PDE5AAPPRAD52KDM4E
SCHEMBL2590586 0.86 SLC2A1 (0.73) SOS1PDE5AEGFRAPPCTNNB1
SCHEMBL2588903 0.85 SOS1 (0.72) SOS1PDE5AAPPRAD52KDM4E
SCHEMBL2588773 0.85 SOS1 (0.66) SOS1PDE5AKDM4EALDH1A1MAPT
SCHEMBL4738601 0.84 RAD52 (0.62) SOS1PDE5AEGFRAPPRAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed