SCHEMBL25890706

SCHEMBL25890706

CNc1ncc(-c2ccc3ccccc3c2)s1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.54
WNT1 P04628 5/20 0.49
DYRK1A Q13627 5/20 0.49
GSK3B P49841 4/20 0.49
KDR P35968 11/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23048870 0.81 DYRK1A (0.64) WNT1DYRK1AGSK3BKDR
SCHEMBL13513650 0.80 KDR (0.66) KDRNPC1RAB9ACYP1A2CYP3A4
SCHEMBL21313815 0.79 ADORA2A (0.49) ARWNT1DYRK1AGSK3BNPC1
SCHEMBL6178573 0.79 KDR (0.70) KDR
Bromide SCHEMBL2527162 0.78 ADORA2A (0.48) ARWNT1DYRK1AGSK3BNPC1
SCHEMBL27631112 0.77 HSD17B1 (0.56) ARNPC1RAB9ACYP1A2CYP3A4
SCHEMBL13680663 0.76 KDR (0.56) KDR
SCHEMBL10013475 0.74 HSD17B1 (0.53) ARNPC1RAB9ACYP1A2CYP3A4
SCHEMBL10013474 0.74 HSD17B1 (0.53) ARNPC1RAB9ACYP1A2CYP3A4
SCHEMBL24112366 0.74 NPC1 (0.44) NPC1RAB9ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3741757-B1 DIHYDROINDOLIZINONE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2023-07-26 EP disclosed