SCHEMBL13680663

SCHEMBL13680663

CNc1ncc(-c2cccc(C)c2)s1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.56
HSD17B1 P14061 2/20 0.49
HSD17B2 P37059 2/20 0.49
KMO O15229 1/20 0.48
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
GSTO1 P78417 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13513650 0.84 KDR (0.66) KDRGSTO1
SCHEMBL3459364 0.80 HSD17B1 (0.54) KDRHSD17B1HSD17B2HDAC1HDAC6
SCHEMBL6180047 0.79 KDR (0.77) KDR
SCHEMBL10079021 0.79 KDR (0.53) KDRHSD17B1HSD17B2HDAC1HDAC6
SCHEMBL9954813 0.77 ALDH1A1 (0.54) KDRHSD17B1HSD17B2HDAC1HDAC6
SCHEMBL12909537 0.77 KDR (0.59) KDRHDAC1HDAC6
SCHEMBL9954919 0.77 HSD17B1 (0.51) KDRHSD17B1HSD17B2HDAC1HDAC6
SCHEMBL25890706 0.76 AR (0.54) KDR
SCHEMBL11965515 0.75 HSD17B1 (0.50) KDRHSD17B1HSD17B2HDAC1HDAC6
SCHEMBL18122016 0.75 HSD17B1 (0.57) KDRHSD17B1HSD17B2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed