SCHEMBL25899638

SCHEMBL25899638

CCn1cc(C(C)=O)c2ccc(C(C)(C)C)nc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.48
CYP1A2 P05177 2/20 0.48
HSD17B10 Q99714 2/20 0.48
KDM4E B2RXH2 2/20 0.48
NFKB1 P19838 1/20 0.48
BLM P54132 1/20 0.48
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
ABCC4 O15439 1/20 0.47
PKM P14618 1/20 0.47
PTGS1 P23219 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.42
TSHR P16473 4/20 0.42
HIF1A Q16665 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 4/20 0.40
MAPK1 P28482 2/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25899951 0.81 KMT2A (0.68) LMNACYP1A2HSD17B10KDM4ENFKB1
SCHEMBL2546290 0.74 CNR1 (0.51)
SCHEMBL12248454 0.72 KMT2A (0.80) LMNACYP1A2HSD17B10KDM4ENFKB1
SCHEMBL11788404 0.72 LMNA (0.70) LMNACYP1A2HSD17B10KDM4ENFKB1
SCHEMBL10193346 0.68 LMNA (0.49) LMNACYP1A2HSD17B10KDM4EMEN1
Trifluoroacetic Acid SCHEMBL12481205 0.67 CFD (0.42) LMNACYP1A2HSD17B10KDM4ENFKB1
SCHEMBL13610849 0.67 KMT2A (0.74) LMNACYP1A2HSD17B10KDM4ENFKB1
SCHEMBL13967354 0.67 CFD (0.44) LMNACYP1A2KDM4EMEN1KMT2A
Nalidixic Acid SCHEMBL9743582 0.66 KMT2A (0.97) LMNACYP1A2HSD17B10KDM4ENFKB1
SCHEMBL17176644 0.66 HTR3A (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138362-A1 WEE1 INHIBITOR, PREPARATION THEREFOR, AND USE THEREOF 江苏天士力帝益药业有限公司 2023-07-27 WO disclosed