Bromide

Bromide

SCHEMBL2590637

Br.CCCCN1c2ccc(Br)cc2Sc2cc(Br)ccc21

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 1/20 0.40
CHRM2 known ✓ P08172 1/20 0.40
HTR1A known ✓ P08908 1/20 0.40
ADRA2A known ✓ P08913 1/20 0.40
ADRA2B known ✓ P18089 1/20 0.40
ADRA2C known ✓ P18825 1/20 0.40
CHRM3 known ✓ P20309 1/20 0.40
SLC6A2 known ✓ P23975 1/20 0.40
ADRA1D known ✓ P25100 1/20 0.40
SLC6A4 known ✓ P31645 1/20 0.40
ADRA1A known ✓ P35348 1/20 0.40
SIGMAR1 known ✓ Q99720 1/20 0.40
DRD2 P14416 2/20 0.50
HTR2A P28223 2/20 0.50
HTR7 P34969 2/20 0.50
HTR6 P50406 2/20 0.50
PRMT1 Q99873 2/20 0.47
KDM1A O60341 3/20 0.46
TSHR P16473 2/20 0.43
ALDH1A1 P00352 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8739350 0.92 DRD2 (0.49) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL31069660 0.92 DRD2 (0.49) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL28344805 0.92 DRD2 (0.49) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL801271 0.92 DRD2 (0.49) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL30501546 0.92 DRD2 (0.49) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL31069659 0.92 DRD2 (0.49) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL20288065 0.92 DRD2 (0.49) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL17419212 0.91 KDM1A (0.58) DRD2HTR2AHTR7HTR6KDM1A
SCHEMBL12073897 0.88 DRD2 (0.53) DRD2HTR2AHTR7HTR6PRMT1
SCHEMBL28593684 0.86 PDF (0.53) DRD2HTR2AHTR7HTR6KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585073-A1 ANTIVIRAL COMPOUNDS Prostetta Antiviral Inc. (US) 2013-05-01 EP disclosed
WO-2011137447-A1 ANTIVIRAL COMPOUNDS PROSTETTA ANTIVIRAL INC. (US) 2011-11-03 WO disclosed