SCHEMBL25916624

SCHEMBL25916624

Cc1nc(N)sc1CC(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 8/20 0.55
HRH1 P35367 2/20 0.55
HRH4 Q9H3N8 2/20 0.55
CYP1A2 P05177 1/20 0.55
NOS1 P29475 1/20 0.45
FBP1 P09467 1/20 0.43
ALDH1A1 P00352 3/20 0.38
HSD17B10 Q99714 2/20 0.38
HPGD P15428 1/20 0.38
PRMT6 Q96LA8 1/20 0.37
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PIK3CG P48736 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24410134 0.82 HRH2 (0.57) HRH2HRH1HRH4CYP1A2NOS1
SCHEMBL5911654 0.80 HRH2 (0.55) HRH2HRH1HRH4CYP1A2NOS1
SCHEMBL13459260 0.77
SCHEMBL1911605 0.74
SCHEMBL259638 0.73 HRH2 (0.68) HRH2HRH1HRH4CYP1A2NOS1
SCHEMBL13458766 0.72
SCHEMBL25916625 0.72 NOS1 (0.45) HRH2HRH1HRH4CYP1A2NOS1
SCHEMBL31661267 0.71 ALDH1A1 (0.60) CYP1A2FBP1ALDH1A1HSD17B10HPGD
SCHEMBL5911593 0.71 HRH2 (0.70) HRH2HRH1HRH4CYP1A2NOS1
Amthamine SCHEMBL400272 0.71 HRH2 (1.00) HRH2HRH1HRH4CYP1A2NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023141262-A1 BAX ACTIVATORS AND USE THEREOF IPSEN PHARMA S.A.S. (FR) 2023-07-27 WO disclosed