SCHEMBL2592593

SCHEMBL2592593

NNC(=O)C1(c2cccnc2)CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
LMNA P02545 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
HDAC4 P56524 3/20 0.49
ITGA4 P13612 2/20 0.46
ITGB7 P26010 2/20 0.46
IDO1 P14902 1/20 0.45
HTT P42858 2/20 0.45
HDAC1 Q13547 2/20 0.45
AKR1C1 Q04828 1/20 0.44
P2RX7 Q99572 2/20 0.43
HSD11B1 P28845 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
VNN1 O95497 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21380384 0.95 ALDH1A1 (0.50) ALDH1A1LMNANPSR1HDAC4ITGA4
SCHEMBL17896072 0.84 AKR1C1 (0.62) ALDH1A1LMNANPSR1HDAC4ITGA4
SCHEMBL25460767 0.84 ALDH1A1 (0.53) ALDH1A1LMNANPSR1HDAC4ITGA4
SCHEMBL3664975 0.83 LMNA (0.47) ALDH1A1LMNANPSR1HDAC4ITGA4
SCHEMBL15823293 0.83 LMNA (0.47) ALDH1A1LMNANPSR1HDAC4ITGA4
SCHEMBL9338162 0.83 AKR1C1 (0.65) ALDH1A1LMNANPSR1HDAC4ITGA4
SCHEMBL89653 0.81 OPRM1 (0.47) ALDH1A1LMNANPSR1HDAC4ITGA4
SCHEMBL18400294 0.81 HDAC4 (0.72) ALDH1A1LMNANPSR1HDAC4HTT
SCHEMBL18400378 0.81 HDAC4 (0.72) ALDH1A1LMNANPSR1HDAC4HTT
SCHEMBL18400386 0.81 HDAC4 (0.72) ALDH1A1LMNANPSR1HDAC4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011134877-A1 HETEROBIARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-03 WO disclosed