SCHEMBL25929255

SCHEMBL25929255

CCc1cc(-c2cnc3c(n2)c(-c2cnn(C4CCN(CC)CC4)c2)cn3S(=O)(=O)c2ccccc2)cnc1N1CCN(C)CC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.36
MET P08581 3/20 0.35
HTR6 P50406 2/20 0.35
KHK P50053 1/20 0.35
ACVR1 Q04771 1/20 0.34
AXL P30530 1/20 0.34
MERTK Q12866 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
GSK3B P49841 1/20 0.33
DYRK1A Q13627 1/20 0.33
BRD4 O60885 1/20 0.33
CNR2 P34972 2/20 0.33
MAP3K5 Q99683 1/20 0.32
JAK1 P23458 1/20 0.32
MAP3K7 O43318 1/20 0.32
TAB1 Q15750 1/20 0.32
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25927780 0.93 JAK2 (0.37) EGFRMETKHKAXLMERTK
SCHEMBL25929553 0.91 BRD4 (0.36) EGFRMETKHKAXLMERTK
SCHEMBL25929297 0.89 HTR6 (0.40) METHTR6ACVR1AXLMERTK
SCHEMBL25927872 0.86 JAK2 (0.38) EGFRMETKHKAXLMERTK
SCHEMBL25931287 0.85 JAK2 (0.42) EGFRMETKHKAXLMERTK
SCHEMBL25929408 0.85 JAK2 (0.36) EGFRMETKHKAXLMERTK
SCHEMBL25929685 0.85 MET (0.34) EGFRMETKHKAXLMERTK
SCHEMBL25927636 0.85 JAK2 (0.35) EGFRMETAXLMERTKPIK3CA
SCHEMBL25929520 0.84 JAK2 (0.36) EGFRMETAXLMERTKPIK3CA
SCHEMBL25931674 0.83 EGFR (0.41) EGFRMETAXLMERTKJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131271-A1 PYRROLE FUSED-RING PYRAZOLE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 杭州中美华东制药有限公司 2023-07-13 WO disclosed