SCHEMBL25930738

SCHEMBL25930738

O=c1c2ccccc2c2ccccc2n1Cc1c2ccccc2cc2c1ccc1ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PGR P06401 2/20 0.43
RORA P35398 2/20 0.43
RORC P51449 2/20 0.43
RORB Q92753 2/20 0.43
TDP1 Q9NUW8 3/20 0.42
HSD17B10 Q99714 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HIF1A Q16665 1/20 0.40
CYP1B1 Q16678 1/20 0.40
NPY5R Q15761 2/20 0.38
HPRT1 P00492 4/20 0.38
BACE1 P56817 1/20 0.37
PAX8 Q06710 1/20 0.37
PARP1 P09874 1/20 0.36
NPC1 O15118 1/20 0.36
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25930731 0.89 PGR (0.50) CYP1A2CYP2C19PGRRORARORC
SCHEMBL25930739 0.84 PGR (0.43) CYP1A2CYP2C9CYP2C19PGRRORA
SCHEMBL25930681 0.83 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19PGRRORA
SCHEMBL25930709 0.80 MCL1 (0.44) CYP1A2CYP2C9CYP2C19PGRRORA
SCHEMBL25930694 0.79 TDP1 (0.49) CYP1A2CYP2C9CYP2C19PGRRORA
SCHEMBL25930678 0.79 PGR (0.47) CYP1A2CYP2C9CYP2C19PGRRORA
SCHEMBL25930717 0.78 PGR (0.43) CYP1A2CYP2C9CYP2C19PGRRORA
SCHEMBL25930705 0.78 PGR (0.43) PGRRORARORCRORBHSD17B10
SCHEMBL25930714 0.77 ALDH1A1 (0.43) CYP1A2CYP2C9CYP2C19PGRRORA
SCHEMBL9405425 0.76 CYP19A1 (0.53) CYP1A2CYP2C19TDP1HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11713319-B2 Compounds having valerolactam structures MERCK PATENT GMBH (DE) 2023-08-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11713319-B2 Compounds having valerolactam structures ACE, CYP3A4, CYP2D6 CYP1A2 32/4885CYP2C9 6/4885CYP2C19 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.