SCHEMBL2593264

SCHEMBL2593264

COC(=O)C1CCCCC1c1noc(C)c1Br

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 1/20 0.41
CPT2 P23786 1/20 0.36
CPT1A P50416 1/20 0.36
EPHX2 P34913 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
BDKRB1 P46663 1/20 0.32
CNR2 P34972 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CHRM2 P08172 1/20 0.30
CHRM4 P08173 1/20 0.30
CHRM3 P20309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2576714 0.75 EPHX2 (0.35) EPHX2SMN1; SMN2KDM4ETDP1
SCHEMBL2576717 0.75 EPHX2 (0.35) EPHX2SMN1; SMN2KDM4ETDP1
SCHEMBL16635759 0.73 SLC6A2 (0.41) SLC6A2SLC6A4CPT2CPT1ASMN1; SMN2
SCHEMBL2593261 0.72 CPT2 (0.48) SLC6A2SLC6A4CPT2CPT1AEPHX2
SCHEMBL17008339 0.71 SLC6A2 (0.45) SLC6A2SLC6A4CPT2CPT1ABDKRB1
SCHEMBL17020281 0.71 SLC6A2 (0.45) SLC6A2SLC6A4CPT2CPT1ABDKRB1
SCHEMBL2595492 0.69 SMN1; SMN2 (0.36) SMN1; SMN2KDM4E
SCHEMBL2596230 0.68 SLC6A2 (0.44) SLC6A2SLC6A4CPT2CPT1ABDKRB1
SCHEMBL16635706 0.67 SLC6A2 (0.36) SLC6A2SLC6A4CPT2CPT1ACNR2
SCHEMBL2595283 0.67 SMN1; SMN2 (0.40) SLC6A2SLC6A4CPT2CPT1ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569319-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F.HOFFMANN-LA ROCHE AG (CH) 2013-03-20 EP disclosed
WO-2011141396-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-17 WO disclosed