SCHEMBL2596230

SCHEMBL2596230

COC(=O)C1CCCCC1c1nnc(C)o1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 1/20 0.44
CPT2 P23786 1/20 0.37
CPT1A P50416 1/20 0.37
PKM P14618 1/20 0.35
ADCY1 Q08828 2/20 0.33
DPP4 P27487 2/20 0.33
DPP8 Q6V1X1 2/20 0.33
DPP7 Q9UHL4 2/20 0.33
BDKRB1 P46663 1/20 0.33
CCR5 P51681 1/20 0.33
HSD11B1 P28845 1/20 0.33
CNR2 P34972 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM3 P20309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2595542 0.81 ALDH1A1 (0.36) ADCY1CCR5HSD11B1
SCHEMBL2593261 0.75 CPT2 (0.48) SLC6A2SLC6A4CPT2CPT1ACHRM2
SCHEMBL408403 0.73 PKM (0.39) PKMADCY1CCR5HSD11B1
SCHEMBL441026 0.73 PKM (0.39) PKMADCY1CCR5HSD11B1
SCHEMBL13595131 0.69 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3
SCHEMBL8058857 0.69 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3
SCHEMBL272354 0.69 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3
SCHEMBL11514730 0.69 CHRM2 (0.48) SLC6A2SLC6A4CHRM2CHRM4CHRM3
SCHEMBL16636099 0.69 SLC6A2 (0.45) SLC6A2SLC6A4CPT2CPT1ABDKRB1
SCHEMBL406761 0.68 PKM (0.40) PKMADCY1DPP4DPP8DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569319-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F.HOFFMANN-LA ROCHE AG (CH) 2013-03-20 EP disclosed
WO-2011141396-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-17 WO disclosed