SCHEMBL25936006

SCHEMBL25936006

FC(F)(F)c1c[nH]c(CC2CCNCC2)n1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 3/20 0.51
CACNA1G O43497 2/20 0.48
HRH3 Q9Y5N1 7/20 0.44
HRH4 Q9H3N8 4/20 0.44
SLC6A4 P31645 5/20 0.41
GBA1 P04062 1/20 0.38
CACNA1C Q13936 1/20 0.35
APP P05067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30720855 0.78 TLR7 (0.35) CACNA1HCACNA1GCACNA1C
SCHEMBL2514697 0.76 HRH3 (0.47) CACNA1HCACNA1GHRH3HRH4SLC6A4
SCHEMBL12798680 0.72 HTR2C (0.46) HRH3HRH4APP
SCHEMBL27324678 0.72 ADRB1 (0.40) HRH3
Hydrochloric Acid SCHEMBL16992579 0.71 HTR2C (0.47) HRH3HRH4APP
SCHEMBL25145833 0.71 CACNA1H (0.44) CACNA1HCACNA1GHRH3HRH4SLC6A4
SCHEMBL25145562 0.70 CACNA1H (0.49) CACNA1HCACNA1GHRH3HRH4SLC6A4
SCHEMBL25145641 0.70 ADRB1 (0.48) CACNA1HCACNA1GHRH3HRH4GBA1
SCHEMBL25146233 0.69 CACNA1H (0.42) CACNA1HCACNA1GHRH3HRH4GBA1
SCHEMBL25145915 0.69 CACNA1H (0.45) CACNA1HCACNA1GHRH3HRH4SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024088922-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF MONOACYLGLYCEROL LIPASE (MAGL) F. HOFFMANN-LA ROCHE AG (CH) 2024-05-02 WO disclosed
WO-2023144160-A1 NEW HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2023-08-03 WO disclosed