SCHEMBL25939712

SCHEMBL25939712

CCOC(=O)c1c(CNC=N)n(C)c2cc(-c3cccc4ccccc34)c(OC3CCCC3)cc12

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
MAPT P10636 2/20 0.38
P4HB P07237 1/20 0.38
KMT2A Q03164 4/20 0.37
KDM4E B2RXH2 4/20 0.37
HTT P42858 1/20 0.36
CASP3 P42574 2/20 0.36
RAD52 P43351 1/20 0.36
PKM P14618 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
ALOX5 P09917 4/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SAE1 Q9UBE0 1/20 0.35
UBA2 Q9UBT2 1/20 0.35
SPR P35270 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25939726 0.89 TSHR (0.39) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25948949 0.88 CASP3 (0.39) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25948972 0.87 TSHR (0.39) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25947077 0.87 TSHR (0.44) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25939770 0.86 TSHR (0.37) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25947076 0.86 TSHR (0.38) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25947610 0.84 TSHR (0.42) TSHRMAPTKMT2AKDM4EHTT
SCHEMBL25948923 0.83 RAD52 (0.38) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25947609 0.83 TSHR (0.36) TSHRMAPTP4HBKMT2AKDM4E
SCHEMBL25951179 0.80 ALOX5 (0.46) KMT2AKDM4ERAD52ALOX5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4209492-A1 COMPOUND FOR TREATING THROMBOTIC DISEASES Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2023-07-12 EP disclosed