SCHEMBL25948949

SCHEMBL25948949

CCOC(=O)c1c(CNC=N)n(C)c2cc(-c3cccc4ccccc34)c(C3CCCC3)cc12

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.39
KDM4E B2RXH2 3/20 0.38
PKM P14618 1/20 0.38
RAD52 P43351 1/20 0.37
TSHR P16473 1/20 0.37
ALOX5 P09917 3/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 2/20 0.36
P4HB P07237 1/20 0.36
SPR P35270 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CACNA1C Q13936 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ELANE P08246 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25939754 0.89 CASP3 (0.39) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25939712 0.88 TSHR (0.39) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25949793 0.87 PKM (0.44) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25947315 0.87 TSHR (0.41) CASP3KDM4EPKMTSHRALOX5
SCHEMBL25939844 0.86 PKM (0.40) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25939765 0.85 KDM4E (0.39) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25947313 0.85 CASP3 (0.38) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25947741 0.83 PKM (0.43) CASP3KDM4EPKMTSHRALOX5
SCHEMBL25949845 0.83 PKM (0.45) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25947211 0.83 PKM (0.42) CASP3KDM4EPKMTSHRALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4209492-A1 COMPOUND FOR TREATING THROMBOTIC DISEASES Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2023-07-12 EP disclosed