SCHEMBL25944899

SCHEMBL25944899

FC(F)(F)c1cnc(Cc2ccc(C3CNC3)cc2)cn1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.37
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
SLC6A3 Q01959 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP3A5 P20815 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25299062 0.76 SLC6A2 (0.47) KDM1AMAOBSLC6A3
SCHEMBL29497057 0.76 SLC6A2 (0.47) KDM1AMAOBSLC6A3
SCHEMBL20757589 0.75 TRPV4 (0.46) KCNH2SLC6A3TAAR1
SCHEMBL31484342 0.75 TRPV4 (0.46) KCNH2SLC6A3TAAR1
SCHEMBL29497099 0.73 SCN9A (0.43) KCNH2
SCHEMBL25295868 0.73 SCN9A (0.43) KCNH2
SCHEMBL23176457 0.68 CHRNB2 (0.40) SLC6A3
SCHEMBL20757258 0.65 HTR2C (0.66)
SCHEMBL20281953 0.65 HRH4 (0.43) KDM1A
SCHEMBL20757967 0.64 HDAC4 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023144160-A1 NEW HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2023-08-03 WO disclosed