SCHEMBL2594565

SCHEMBL2594565

Ic1ccc2nccc(Nc3n[nH]c4ccccc34)c2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RIPK2 O43353 5/20 0.49
CCNC P24863 2/20 0.48
CDK8 P49336 2/20 0.48
GAK O14976 2/20 0.47
KCNH2 Q12809 2/20 0.47
LCK P06239 1/20 0.47
TGFBR1 P36897 1/20 0.47
MAPK14 Q16539 1/20 0.47
RIPK3 Q9Y572 1/20 0.47
COQ8A Q8NI60 1/20 0.46
NLK Q9UBE8 1/20 0.46
FADS1 O60427 2/20 0.43
ADRA2A P08913 2/20 0.43
ULK1 O75385 1/20 0.43
TRPA1 O75762 1/20 0.43
RAF1 P04049 6/20 0.43
BRAF P15056 6/20 0.43
GRM4 Q14833 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14717834 0.84 RIPK2 (0.69) RIPK2CCNCCDK8GAKKCNH2
SCHEMBL599871 0.79 RIPK2 (0.64) RIPK2CCNCCDK8GAKKCNH2
SCHEMBL12180823 0.78 RIPK2 (0.51) RIPK2GAKKCNH2LCKTGFBR1
SCHEMBL2593012 0.78 RIPK2 (0.77) RIPK2GAKKCNH2LCKTGFBR1
SCHEMBL2595976 0.78 RIPK2 (0.77) RIPK2GAKKCNH2LCKTGFBR1
SCHEMBL17059502 0.73 RIPK2 (0.54) RIPK2GAKKCNH2LCKTGFBR1
SCHEMBL18274872 0.69 TRPA1 (0.57) FADS1ADRA2ATRPA1GRM4
SCHEMBL7346388 0.68 TRPA1 (0.69) TGFBR1MAPK14FADS1ADRA2ATRPA1
SCHEMBL17552302 0.67 RIPK2 (0.70) RIPK2GAKKCNH2LCKTGFBR1
SCHEMBL516494 0.66 FADS1 (0.57) FADS1ADRA2AULK1TRPA1GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011140442-A1 AMINO-QUINOLINES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2011-11-10 WO disclosed