SCHEMBL25947756

SCHEMBL25947756

COc1ccc2cc(CO)c(Cl)nc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 1.00
KDM4E B2RXH2 6/20 1.00
GFER P55789 1/20 0.75
L3MBTL1 Q9Y468 4/20 0.56
KMT2A Q03164 3/20 0.56
NPC1 O15118 4/20 0.52
RAB9A P51151 4/20 0.52
NPSR1 Q6W5P4 2/20 0.46
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
MAPK1 P28482 2/20 0.43
TSHR P16473 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 2/20 0.41
CLK1 P49759 2/20 0.41
HSD17B10 Q99714 2/20 0.41
TP53 P04637 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1886013 0.88 KDM4E (0.78) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL14065435 0.83 ALDH1A1 (0.78) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL1574696 0.83 KDM4E (0.70) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL7147155 0.81 ALDH1A1 (0.68) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL7076958 0.79 ALDH1A1 (0.65) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL8644046 0.79 KMT2A (0.73) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL30908421 0.79 KMT2A (0.73) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL16047420 0.78 ALDH1A1 (0.64) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL27581989 0.78 KDM4E (0.64) ALDH1A1KDM4EGFERL3MBTL1KMT2A
SCHEMBL18571753 0.78 ALDH1A1 (0.66) ALDH1A1KDM4EGFERL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024059186-A1 N-((ISOQUINOLIN-6-YL)METHYL)-1H-PYRAZOLE-4-CARBOXAMID DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS FOR THE TREATMENT OF HEREDITARY ANGIOEDEMA TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-03-21 WO disclosed
EP-3719010-B1 AROMATIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF SICHUAN KELUN BIOTECH BIOPHARMACEUTICAL CO LTD (CN) 2023-07-26 EP disclosed