SCHEMBL25949845

SCHEMBL25949845

CCOC(=O)c1c(CNC)n(C)c2cc(C3CC3)c(-c3cccc4ccccc34)cc12

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.45
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RAD52 P43351 1/20 0.40
CACNA1C Q13936 1/20 0.40
ALOX5 P09917 5/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 2/20 0.39
P4HB P07237 1/20 0.39
SPR P35270 1/20 0.38
CASP3 P42574 1/20 0.38
TSHR P16473 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25949793 0.97 PKM (0.44) PKMKDM4EMAPTNPSR1RAD52
SCHEMBL25939889 0.90 PKM (0.41) PKMKDM4EMAPTNPSR1RAD52
SCHEMBL25947900 0.89 PKM (0.44) PKMKDM4EMAPTNPSR1CACNA1C
SCHEMBL25939844 0.87 PKM (0.40) PKMKDM4EMAPTNPSR1RAD52
SCHEMBL25939765 0.86 KDM4E (0.39) PKMKDM4EMAPTNPSR1RAD52
SCHEMBL25947741 0.86 PKM (0.43) PKMKDM4EMAPTNPSR1CACNA1C
SCHEMBL25947211 0.86 PKM (0.42) PKMKDM4EMAPTNPSR1CACNA1C
SCHEMBL25949826 0.85 RAD52 (0.50) PKMKDM4EMAPTRAD52ALOX5
SCHEMBL25948972 0.85 TSHR (0.39) PKMKDM4EMAPTRAD52ALOX5
SCHEMBL25948907 0.84 RAD52 (0.48) PKMKDM4EMAPTRAD52ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4209492-A1 COMPOUND FOR TREATING THROMBOTIC DISEASES Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2023-07-12 EP disclosed