SCHEMBL25947741

SCHEMBL25947741

CCOC(=O)c1c(CN)n(C)c2cc(C3CCCC3)c(-c3cccc4ccccc34)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.41
CASP3 P42574 2/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CACNA1C Q13936 1/20 0.40
ALOX5 P09917 5/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ELANE P08246 1/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25947315 0.96 TSHR (0.41) PKMTSHRCASP3MAPTNPSR1
SCHEMBL25947900 0.96 PKM (0.44) PKMTSHRCASP3MAPTNPSR1
SCHEMBL25947211 0.93 PKM (0.42) PKMTSHRCASP3MAPTNPSR1
SCHEMBL25949793 0.90 PKM (0.44) PKMTSHRCASP3MAPTNPSR1
SCHEMBL25939844 0.88 PKM (0.40) PKMTSHRCASP3MAPTNPSR1
SCHEMBL25951709 0.87 PKM (0.39) PKMTSHRCASP3MAPTNPSR1
SCHEMBL25947610 0.86 TSHR (0.42) PKMTSHRCASP3MAPTALOX5
SCHEMBL25949845 0.86 PKM (0.45) PKMTSHRCASP3MAPTNPSR1
SCHEMBL25947077 0.84 TSHR (0.44) PKMTSHRCASP3MAPTALOX5
SCHEMBL25947856 0.83 TSHR (0.49) PKMTSHRMAPTNPSR1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4209492-A1 COMPOUND FOR TREATING THROMBOTIC DISEASES Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2023-07-12 EP disclosed