SCHEMBL2596695

SCHEMBL2596695

CCc1cc(-c2nnc(S)n2-c2ccc3[nH]c(C)c(CC)c3c2)c(O)cc1O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.37
HSD17B10 Q99714 2/20 0.37
MAPT P10636 7/20 0.34
GAA P10253 6/20 0.34
KDM4E B2RXH2 5/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
ALDH1A1 P00352 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HTR1D P28221 1/20 0.34
MAPK1 P28482 1/20 0.34
HTR7 P34969 1/20 0.34
HTR3A P46098 1/20 0.34
HTR6 P50406 1/20 0.34
HSP90AA1 P07900 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL421071 0.92 ALDH1A1 (0.38) SMN1; SMN2HSD17B10MAPTKDM4EMEN1
SCHEMBL1586060 0.88 GAA (0.35) MAPTGAAKDM4EMEN1KMT2A
SCHEMBL10345296 0.86 ALDH1A1 (0.37) SMN1; SMN2HSD17B10MAPTKDM4EMEN1
SCHEMBL9924955 0.84 HSP90AA1 (0.34) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL930153 0.83 HSP90AA1 (0.34) SMN1; SMN2MAPTGAAKDM4EMEN1
SCHEMBL15940226 0.82 MAP3K11 (0.39) SMN1; SMN2MAPTGAAKDM4EMEN1
SCHEMBL3701216 0.81 MAPT (0.35) HSD17B10MAPTGAAKDM4EMEN1
SCHEMBL931175 0.80 HTR1A (0.34) SMN1; SMN2MAPTGAAKDM4EALDH1A1
SCHEMBL12694836 0.80 MAP3K11 (0.39) MAPTGAAKDM4EHSP90AA1HSP90AB1
SCHEMBL13983495 0.80 HSP90AA1 (0.33) MAPTGAAKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO claimed