SCHEMBL25968161

SCHEMBL25968161

Cc1cc(F)c(N2CCC(O)(COc3ccc(C)c4c3OCC(=O)N4)CC2)c(F)c1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 8/20 0.33
DRD2 P14416 7/20 0.33
DRD4 P21917 5/20 0.33
HTR1A P08908 4/20 0.31
HTR1D P28221 4/20 0.31
HTR1B P28222 4/20 0.31
HTR7 P34969 3/20 0.31
HTR2A P28223 4/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
BRD4 O60885 1/20 0.31
DRD1 P21728 1/20 0.31
NR3C2 P08235 1/20 0.31
ADRB1 P08588 2/20 0.30
HTR2C P28335 2/20 0.30
MCHR1 Q99705 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20597459 0.84 TRPV4 (0.35) DRD3DRD2DRD4HTR1AHTR1D
SCHEMBL25968118 0.78 HSP90AA1 (0.36) HSP90AA1HSP90AB1
SCHEMBL25969105 0.74 MGLL (0.44) DRD3DRD2HTR1AHTR1DHTR1B
SCHEMBL25970553 0.74 HSP90AA1 (0.33) HTR1AHTR1DHTR1BHSP90AA1HSP90AB1
SCHEMBL20597104 0.71 MGLL (0.33) DRD3DRD2HTR1AHTR1DHTR1B
SCHEMBL20597385 0.71 TRPV4 (0.37)
SCHEMBL17544184 0.71 TRPV4 (0.33)
SCHEMBL20597030 0.70 TRPV4 (0.37) HSP90AA1HSP90AB1
SCHEMBL17542742 0.70 TRPV4 (0.34) HSP90AA1HSP90AB1
SCHEMBL17542937 0.70 TRPV4 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3421454-B9 PIPERIDINE DERIVATIVE OTSUKA PHARMA CO LTD (JP) 2023-08-09 EP disclosed