SCHEMBL2597134

SCHEMBL2597134

CCCC(=O)CS(=O)(=O)Nn1c(=O)[nH]c2cc(CC)c(-c3ccnn3C)cc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.33
PDPK1 O15530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2599232 0.89 LIPG (0.35) HAVCR2
SCHEMBL1663156 0.85 HAVCR2 (0.35) HAVCR2PDPK1
SCHEMBL14719753 0.85 LIPG (0.34) HAVCR2
SCHEMBL1661264 0.78 HAVCR2 (0.34) HAVCR2
SCHEMBL2597135 0.77 HAVCR2 (0.32) HAVCR2
SCHEMBL4628060 0.76 HAVCR2 (0.33) HAVCR2
Benzoylenurea SCHEMBL15948987 0.76 KDM4E (0.34) HAVCR2PDPK1
SCHEMBL14719786 0.76 CD274 (0.36)
SCHEMBL1661316 0.75 USP1 (0.32) HAVCR2
SCHEMBL1660973 0.75 CCNK (0.37) HAVCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571865-A1 2,4-DIOXO-1,4-DIHYDRO-2H-QUINAZOLIN-3-YL-SULFONAMIDE DERIVATIVES Novartis AG (CH) 2013-03-27 EP disclosed
WO-2011144666-A1 2,4-DIOXO-1,4-DIHYDRO-2H-QUINAZOLIN-3-YL-SULFONAMIDE DERIVATIVES NOVARTIS AG (CH) 2011-11-24 WO disclosed