SCHEMBL2597583

SCHEMBL2597583

N#Cc1c(F)ccc(Nc2ncc(Oc3cccc(N4CCOCC4)c3)cn2)c1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 2/20 0.44
CDK2 P24941 2/20 0.44
CDK9 P50750 2/20 0.44
CCNE1 P24864 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
F10 P00742 1/20 0.41
NTRK1 P04629 2/20 0.40
RIPK2 O43353 1/20 0.40
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNA2 P20248 1/20 0.39
CDK7 P50613 1/20 0.39
CCNH P51946 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2597767 0.90 CCNT1 (0.42) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL2597549 0.87 CCNT1 (0.43) CCNT1CDK2CDK9CCNE1KDM4E
SCHEMBL2597649 0.86 CCNT1 (0.45) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL31054180 0.82 CCNT1 (0.52) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL2597569 0.82 CCNT1 (0.52) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL2597604 0.79 CCNT1 (0.47) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL2597598 0.78 HDAC3 (0.53) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL2598615 0.75 JAK2 (0.45) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL2597585 0.75 HDAC3 (0.48) CCNT1CDK2CDK9CCNE1HDAC3
SCHEMBL3655248 0.73 TYK2 (0.46) F10GSK3ALRRK2MAPK15CAMKK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP claimed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO claimed
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed