SCHEMBL2598615

SCHEMBL2598615

COc1ccc(Nc2ncc(Oc3cccc(N4CCOCC4)c3)cn2)cc1C#N.N#Cc1cc(Nc2ncc(Oc3cccc(N4CCCC4)c3)cn2)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.45
TBK1 Q9UHD2 5/20 0.45
CDK2 P24941 5/20 0.44
CCNT1 O60563 4/20 0.44
CDK9 P50750 4/20 0.44
CCNE1 P24864 2/20 0.44
RIPK2 O43353 1/20 0.43
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
CSF1R P07333 3/20 0.41
GALR2 O43603 1/20 0.41
GALR1 P47211 1/20 0.41
LCK P06239 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2597630 0.93 JAK2 (0.51) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL31054180 0.91 CCNT1 (0.52) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL2597569 0.91 CCNT1 (0.52) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL2597608 0.88 CCNT1 (0.47) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL2597585 0.81 HDAC3 (0.48) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL2597767 0.78 CCNT1 (0.42) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL2597598 0.77 HDAC3 (0.53) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL2597549 0.76 CCNT1 (0.43) JAK2TBK1CDK2CCNT1CDK9
SCHEMBL2597649 0.76 CCNT1 (0.45) JAK2CDK2CCNT1CDK9CCNE1
SCHEMBL2597604 0.76 CCNT1 (0.47) JAK2TBK1CDK2CCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed