SCHEMBL2597585

SCHEMBL2597585

N#Cc1cc(Nc2ncc(Oc3cccc(N4CCOCC4)c3)cn2)ccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
PKMYT1 Q99640 1/20 0.46
NTRK1 P04629 2/20 0.46
JAK2 O60674 3/20 0.46
TBK1 Q9UHD2 2/20 0.46
CCNT1 O60563 2/20 0.45
CDK2 P24941 2/20 0.45
CDK9 P50750 2/20 0.45
CCNE1 P24864 1/20 0.45
CCNA2 P20248 1/20 0.45
BRD4 O60885 1/20 0.44
MAP3K7 O43318 1/20 0.44
MAPK1 P28482 1/20 0.44
MAP2K1 Q02750 1/20 0.44
PLK1 P53350 1/20 0.43
EPHB4 P54760 1/20 0.43
PLA2G7 Q13093 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2597767 0.89 CCNT1 (0.42) HDAC3HDAC1HDAC2HDAC6PKMYT1
SCHEMBL2597569 0.89 CCNT1 (0.52) HDAC3HDAC1HDAC2HDAC6NTRK1
SCHEMBL31054180 0.89 CCNT1 (0.52) HDAC3HDAC1HDAC2HDAC6NTRK1
SCHEMBL2597630 0.87 JAK2 (0.51) HDAC3HDAC1HDAC2HDAC6PKMYT1
SCHEMBL2597598 0.84 HDAC3 (0.53) HDAC3HDAC1HDAC2HDAC6NTRK1
SCHEMBL2598615 0.81 JAK2 (0.45) HDAC3HDAC1HDAC2HDAC6JAK2
SCHEMBL2597549 0.80 CCNT1 (0.43) HDAC3HDAC1HDAC2HDAC6NTRK1
SCHEMBL2597608 0.80 CCNT1 (0.47) HDAC3HDAC1HDAC2HDAC6JAK2
SCHEMBL2597604 0.79 CCNT1 (0.47) HDAC3HDAC1HDAC2HDAC6NTRK1
SCHEMBL2597597 0.76 DHFR (0.45) HDAC3HDAC1HDAC2HDAC6NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP claimed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO claimed
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed