SCHEMBL25975830

SCHEMBL25975830

Cc1cnc2c(c1)CN(CCCF)CC2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.40
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 2/20 0.38
POLB P06746 1/20 0.37
ABCB1 P08183 1/20 0.36
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25975832 0.82 PDCD1 (0.42) LMNAMAPTTP53ADORA2AADORA1
SCHEMBL14566140 0.80 ADORA2A (0.40) LMNAMAPTTP53ADORA2AADORA1
SCHEMBL14566143 0.80 CDK4 (0.41) LMNAMAPTTP53ADORA2AADORA1
SCHEMBL25975828 0.78 CDK4 (0.38) LMNAMAPTTP53ADORA2AADORA1
SCHEMBL26032299 0.78 POLB (0.41) LMNAMAPTTP53ADORA2AADORA1
SCHEMBL18098800 0.78 ADORA2A (0.39) LMNAMAPTTP53ADORA2AADORA1
SCHEMBL14853093 0.77 CYP2C19 (0.45) LMNAMAPTADORA2AADORA1POLB
SCHEMBL14853336 0.75 HRH3 (0.37) LMNAADORA2AADORA1POLBDRD2
SCHEMBL14853095 0.73 MEN1 (0.60) LMNAMAPTTP53MEN1KMT2A
SCHEMBL22739185 0.72 ADORA2A (0.33) LMNAADORA2AADORA1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154282-A1 COMPOUNDS HAVING A T-STRUCTURE FORMED BY AT LEAST FOUR CYCLES FOR USE IN THE TREATMENT OF CANCER AND OTHER INDICATIONS THERAS, INC. (US) 2023-08-17 WO disclosed