SCHEMBL2597600

SCHEMBL2597600

N#Cc1cc(Nc2ncc(O)cn2)ccc1F

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SYK P43405 7/20 0.49
AURKA O14965 4/20 0.49
GRM4 Q14833 1/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.43
VNN1 O95497 1/20 0.41
GRM5 P41594 1/20 0.41
KDR P35968 1/20 0.40
CCNT1 O60563 2/20 0.38
CCNA2 P20248 2/20 0.38
CDK2 P24941 2/20 0.38
CDK9 P50750 2/20 0.38
CCNA1 P78396 2/20 0.38
BLM P54132 1/20 0.38
WRN Q14191 1/20 0.38
EGFR P00533 1/20 0.37
ERBB2 P04626 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2597599 0.79 MAOB (0.47) SYKGRM4ABCG2KDRCDK2
SCHEMBL655595 0.74 SYK (0.64) SYKAURKAKDRCDK2
SCHEMBL2597602 0.74 KDR (0.44) SYKGRM4ABCG2KDREGFR
SCHEMBL19190440 0.72 GRM4 (0.50) GRM4ABCG2VNN1BLMWRN
SCHEMBL1198249 0.72 SYK (0.59) SYKAURKAKDRCDK2
SCHEMBL24127052 0.71 ABCG2 (0.56) GRM4ABCG2
SCHEMBL4006335 0.70 SYK (0.49) SYKAURKAGRM4ABCG2EGFR
SCHEMBL26186327 0.70 GRM4 (0.47) GRM4ABCG2KDRBLMWRN
SCHEMBL3173181 0.70 GRM4 (0.48) GRM4ABCG2BLMWRNEGFR
SCHEMBL189517 0.69 ESR1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed