SCHEMBL2598341

SCHEMBL2598341

CC(O)Cn1ncc2ncc(F)c(Cl)c21

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 3/20 0.42
HTR2A P28223 5/20 0.37
HTR2C P28335 5/20 0.37
HTR2B P41595 3/20 0.37
GRIN2B Q13224 2/20 0.31
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
MAP2K1 Q02750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2598339 1.00 TGFBR1 (0.42) TGFBR1HTR2AHTR2CHTR2BGRIN2B
SCHEMBL2598395 0.80 TGFBR1 (0.37) TGFBR1GRIN2BLMNA
SCHEMBL2598413 0.77 LRRK2 (0.39) GRIN2BSMN1; SMN2
SCHEMBL2598340 0.74 TGFBR1 (0.46) TGFBR1GRIN2B
SCHEMBL2596838 0.70 TGFBR1 (0.44) TGFBR1
SCHEMBL22119118 0.67 EGLN1 (0.36) TGFBR1HTR2AHTR2CHTR2BLMNA
SCHEMBL22119121 0.67 EGLN1 (0.36) TGFBR1HTR2AHTR2CHTR2BLMNA
SCHEMBL22119590 0.67 HTR2A (0.40) TGFBR1HTR2AHTR2CHTR2B
SCHEMBL22118993 0.67 HTR2A (0.40) TGFBR1HTR2AHTR2CHTR2B
SCHEMBL25320454 0.62 CSNK2A1 (0.38) HTR2AHTR2CHTR2BLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146287-A1 PYRAZOLO[4,3-B]PYRIDINE-7-AMINE INHIBITORS OF ALK5 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-11-24 WO disclosed