SCHEMBL2598922

SCHEMBL2598922

O=C(O)N1CC2CCOc3c(Cl)cccc3[C@H]2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
ADRA1A P35348 1/20 0.39
NOTUM Q6P988 3/20 0.38
HSD11B1 P28845 2/20 0.37
TDP1 Q9NUW8 1/20 0.35
CNR1 P21554 1/20 0.35
ATM Q13315 1/20 0.34
PSMB8 P28062 2/20 0.33
PSMB5 P28074 1/20 0.33
CCR5 P51681 1/20 0.32
P2RX7 Q99572 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1806180 1.00 ADRA2A (0.39) ADRA2AADRA2BADRA2CADRA1ANOTUM
SCHEMBL1806181 1.00 ADRA2A (0.39) ADRA2AADRA2BADRA2CADRA1ANOTUM
SCHEMBL1806059 1.00 ADRA2A (0.39) ADRA2AADRA2BADRA2CADRA1ANOTUM
SCHEMBL1806062 1.00 ADRA2A (0.39) ADRA2AADRA2BADRA2CADRA1ANOTUM
SCHEMBL1806058 1.00 ADRA2A (0.39) ADRA2AADRA2BADRA2CADRA1ANOTUM
SCHEMBL1804905 0.86 ACHE (0.40) HSD11B1
SCHEMBL1804909 0.86 ACHE (0.40) HSD11B1
SCHEMBL2599017 0.86 ACHE (0.40) HSD11B1
SCHEMBL1804907 0.86 ACHE (0.40) HSD11B1
SCHEMBL1802527 0.85 ADRA2A (0.39) ADRA2AADRA1ANOTUMHSD11B1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571353-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF AbbVie Inc. (US) 2013-03-27 EP disclosed
WO-2011146089-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2011-11-24 WO disclosed