SCHEMBL2599647

SCHEMBL2599647

Fc1cccc2c1OCC=N2

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.38
SYK P43405 1/20 0.33
CYP19A1 P11511 2/20 0.31
TERT O14746 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1029989 0.77 ADRA2A (0.37) ADRA2A
SCHEMBL2635508 0.72 TRPA1 (0.39)
SCHEMBL1649469 0.70 TRPA1 (0.50)
SCHEMBL30403098 0.70 CA2 (0.36)
SCHEMBL224636 0.67 TRPA1 (0.42) SYK
Ammonia Solution, Strong SCHEMBL28509301 0.65 TRPA1 (0.41) SYK
Hydrochloric Acid SCHEMBL7159867 0.65 TRPA1 (0.41) SYK
SCHEMBL30794527 0.65
SCHEMBL8191555 0.63 CA2 (0.40) ADRA2ACYP19A1TERT
SCHEMBL16430044 0.63 CA12 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed