SCHEMBL26005804

SCHEMBL26005804

O=Cc1cc(F)ccc1-n1cc(Br)c2ccncc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
IDO1 P14902 2/20 0.35
MAPT P10636 4/20 0.34
HTT P42858 2/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CHUK O15111 1/20 0.33
ROCK2 O75116 1/20 0.32
DYRK1A Q13627 2/20 0.32
NFATC1 O95644 1/20 0.32
GSK3B P49841 1/20 0.32
ACHE P22303 2/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
SCN9A Q15858 1/20 0.31
KDR P35968 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19972684 0.82 KDM4C (0.40) ALDH1A1IDO1GAAKDM4C
SCHEMBL26006720 0.79 DRD2 (0.36) ALDH1A1KDM4EIDO1KDM4C
SCHEMBL25135361 0.78 KDM4E (0.33) ALDH1A1KDM4E
SCHEMBL25135242 0.77 KCNH2 (0.42)
SCHEMBL19972556 0.76 KDM4C (0.33) IDO1ROCK2SCN9AKDM4C
SCHEMBL19980679 0.75 PTGDR2 (0.35) ALDH1A1KDM4E
SCHEMBL19980726 0.74 HTR6 (0.39)
SCHEMBL26005471 0.73 DRD2 (0.37) ALDH1A1KDM4EDYRK1A
SCHEMBL19980734 0.73 KDM4C (0.31) KDM4C
SCHEMBL25135199 0.72 HRH2 (0.43) ALDH1A1ROCK2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4230627-A2 INHIBITORS OF THE MENIN-MLL INTERACTION Vitae Pharmaceuticals, LLC (US) 2023-08-23 EP disclosed