SCHEMBL26017113

SCHEMBL26017113

CC(C)N(I)Cc1ccc(C2(C(F)(F)F)CC2)cc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.33
PDE2A O00408 3/20 0.33
EPHX2 P34913 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
WDR5 P61964 1/20 0.31
CACNA1H O95180 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26036976 0.77 MEN1 (0.33) SIGMAR1PDE2AEPHX2NR1H4CACNA1H
SCHEMBL26014791 0.76 PTGS1 (0.40) SIGMAR1PDE2A
SCHEMBL26017234 0.73 SLC6A2 (0.30)
SCHEMBL19302498 0.73 SIGMAR1 (0.39) SIGMAR1EPHX2NR1H4CACNA1H
SCHEMBL24196137 0.70 PDK2 (0.39) SIGMAR1CACNA1H
SCHEMBL19275237 0.70 PDE2A (0.42) SIGMAR1PDE2AEPHX2NR1H4
SCHEMBL21035484 0.70 CACNA1H (0.36) SIGMAR1EPHX2NR1H4WDR5CACNA1H
SCHEMBL21036238 0.70 PDK2 (0.37) SIGMAR1EPHX2NR1H4WDR5CACNA1H
SCHEMBL24196140 0.70 LOXL2 (0.41) SIGMAR1CACNA1H
SCHEMBL25735734 0.69 PDK2 (0.40) SIGMAR1EPHX2NR1H4CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154291-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed