SCHEMBL260408

SCHEMBL260408

O=Cc1ccc(Oc2cccc(Br)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
MAOB P27338 3/20 0.49
MAOA P21397 2/20 0.49
SMN1; SMN2 Q16637 3/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 1/20 0.47
PARP10 Q53GL7 1/20 0.46
PARP3 Q9Y6F1 1/20 0.46
PGR P06401 1/20 0.43
MAPT P10636 3/20 0.43
CHEK1 O14757 1/20 0.43
KDR P35968 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CASP3 P42574 1/20 0.43
HTT P42858 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
CYP2A6 P11509 1/20 0.42
TTR P02766 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5216508 0.87 ALDH1A1 (0.68) ALDH1A1MAOBMAOASMN1; SMN2LMNA
SCHEMBL8546955 0.87 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2KDM4ELMNAPARP10
SCHEMBL3839157 0.84 ALDH1A1 (0.54) ALDH1A1MAOBSMN1; SMN2PGRMAPT
SCHEMBL3838974 0.84 ALDH1A1 (0.54) ALDH1A1MAOBSMN1; SMN2PGRMAPT
SCHEMBL6853633 0.83 SRC (0.53) ALDH1A1MAOBMAOASMN1; SMN2KDM4E
SCHEMBL31599170 0.83 SRC (0.53) ALDH1A1MAOBMAOASMN1; SMN2KDM4E
SCHEMBL3838956 0.82 SMN1; SMN2 (0.58) ALDH1A1MAOBSMN1; SMN2LMNAPGR
SCHEMBL7936134 0.82 MAOA (0.62) ALDH1A1MAOBMAOASMN1; SMN2LMNA
SCHEMBL28642171 0.81 MAOB (0.56) ALDH1A1MAOBMAOASMN1; SMN2KDM4E
SCHEMBL260494 0.81 PARP10 (0.55) ALDH1A1MAOBMAOASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103070854-A Fused ring compound TAKEDA PHARMACEUTICAL 2013-05-01 CN disclosed
CN-101616913-B Fused ring compound TAKAEDA CHEMICAL IND LTD 2013-01-23 CN disclosed
CN-102731451-A Fused ring compound TAKEDA PHARMACEUTICAL 2012-10-17 CN disclosed
US-8067440-B2 Phosphonium salts derivatives and uses thereof VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-11-29 US disclosed
US-8067440-B2 Phosphonium salts derivatives and uses thereof VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-11-29 US disclosed
US-20110092683-A1 PHOSPHONIUM SALTS DERIVATIVES AND USES THEREOF VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-04-21 US disclosed
US-20110092683-A1 PHOSPHONIUM SALTS DERIVATIVES AND USES THEREOF VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-04-21 US disclosed
US-7880037-B2 Phosphonium supported triphenylphosphine; for controlling solubility of a molecule; oxidation of Cinnamyl Alcohol using above catalyst system VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-02-01 US disclosed
US-7880037-B2 Phosphonium supported triphenylphosphine; for controlling solubility of a molecule; oxidation of Cinnamyl Alcohol using above catalyst system VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-02-01 US disclosed
CN-101616913-A Fused ring compound TAKEDA PHARMACEUTICAL 2009-12-30 CN disclosed
US-20070197477-A1 PHOSPHONIUM SALTS DERIVATIVES VALORISATION-RECHERECHE (CA) 2007-08-23 US disclosed
US-20070197477-A1 PHOSPHONIUM SALTS DERIVATIVES VALORISATION-RECHERECHE (CA) 2007-08-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070197477-A1 PHOSPHONIUM SALTS DERIVATIVES PI4K2A, PIP4K2A, PI4K2B ALDH1A1 3806/4885MAOB 2765/4885MAOA 2081/4885
US-20110092683-A1 PHOSPHONIUM SALTS DERIVATIVES AND USES THEREOF PI4K2A, PIP4K2A, PI4K2B ALDH1A1 3468/4885MAOB 2010/4885MAOA 1675/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.