SCHEMBL260601

SCHEMBL260601

CCCC(CCC)C(=O)Nc1nc(C)c(CCO[N+](=O)[O-])s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 4/20 0.40
PSEN2 P49810 4/20 0.40
APH1B Q8WW43 4/20 0.40
NCSTN Q92542 4/20 0.40
APH1A Q96BI3 4/20 0.40
PSENEN Q9NZ42 4/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
POLB P06746 2/20 0.35
RXFP1 Q9HBX9 2/20 0.34
CYP1A2 P05177 1/20 0.34
GAA P10253 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
ALDH1A1 P00352 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL260907 0.82 ALDH1A1 (0.46) POLBMEN1KMT2AITGB3ITGA2B
SCHEMBL264227 0.80 MAPT (0.43) POLBRXFP1GAATSHRSMN1; SMN2
SCHEMBL261252 0.79 ITGB3 (0.33) GAASMN1; SMN2MEN1KMT2AITGB3
SCHEMBL260758 0.79 ATAD2 (0.43) RXFP1GAASMN1; SMN2MEN1KMT2A
SCHEMBL264106 0.78
SCHEMBL12590840 0.78 MEN1 (0.31) GAAMEN1KMT2A
SCHEMBL260360 0.78 ALDH1A1 (0.31) CYP1A2GAASMN1; SMN2MEN1KMT2A
SCHEMBL261256 0.78 GAA (0.31) CYP1A2GAASMN1; SMN2MEN1KMT2A
SCHEMBL260339 0.78 ITGB3 (0.43) TSHRSMN1; SMN2MEN1KMT2AITGB3
SCHEMBL261174 0.77 ALDH1A1 (0.33) GAAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134010-B2 4-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-phenylamine; N-{4-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-phenyl}-acetamide; or4-Methyl-5-(2-nitrooxy-ethyl)-2-(4-nitro-phenyl)-thiazole; cardiovascular, gastrointestinal, inflammatory, respiratory disease RENOPHARM LTD. (IL) 2012-03-13 US disclosed