SCHEMBL2606325

SCHEMBL2606325

COc1ccc(C2(O)c3ccc(O[Si](C)(C)C(C)(C)C)cc3OCC2c2ccc(CC(C)(C)[Si](C)(C)O)cc2)cc1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.32
ALOX12 P18054 2/20 0.32
SCN9A Q15858 1/20 0.31
KCNH2 Q12809 1/20 0.30
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL240709 0.89 ALOX15 (0.37) ALOX15ALOX12KCNH2TRPV1
SCHEMBL12062893 0.84
SCHEMBL2570841 0.79 ALOX15 (0.44) ALOX15ALOX12KCNH2TRPV1
SCHEMBL15966183 0.77 DRD2 (0.31)
SCHEMBL12162878 0.76
SCHEMBL245775 0.76 ALOX15 (0.31) ALOX15ALOX12
SCHEMBL2570060 0.75 ALOX15 (0.44) ALOX15ALOX12KCNH2TRPV1
SCHEMBL2606319 0.75 CYP19A1 (0.47) ALOX15ALOX12KCNH2TRPV1
SCHEMBL10042945 0.74 ALOX12 (0.42) ALOX15ALOX12KCNH2TRPV1
SCHEMBL12052438 0.73 ALOX12 (0.41) ALOX15ALOX12KCNH2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160136129-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2016-05-19 US disclosed
US-9198895-B2 Chroman derivatives, medicaments and use in therapy MEI PHARMA, INC. (US) 2015-12-01 US disclosed
US-20150238458-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2015-08-27 US disclosed
US-8957109-B2 Chroman derivatives, medicaments and use in therapy MEI PHARMA, INC. (US) 2015-02-17 US disclosed
US-20140161908-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MEI PHARMA, INC. (US) 2014-06-12 US disclosed
US-8461361-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2013-06-11 US disclosed
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-07-05 US disclosed
US-8163795-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2012-04-24 US disclosed
US-20120004296-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC (US) 2012-01-05 US disclosed
US-8080675-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2011-12-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150238458-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 3665/4885ALOX12 3724/4885SCN9A 4828/4885
US-20160136129-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 3665/4885ALOX12 3724/4885SCN9A 4828/4885
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 3665/4885ALOX12 3724/4885SCN9A 4828/4885
US-20140161908-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 4133/4885ALOX12 4083/4885SCN9A 4849/4885
US-20120004296-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 3665/4885ALOX12 3724/4885SCN9A 4828/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.