SCHEMBL2610140

SCHEMBL2610140

Cc1ccccc1C(C#N)O[Si](C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.42
TSHR P16473 2/20 0.35
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SGMS2 Q8NHU3 2/20 0.33
ADRA2A P08913 2/20 0.33
ADRA2B P18089 2/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
ADRA2C P18825 1/20 0.33
CYP19A1 P11511 1/20 0.33
GAA P10253 1/20 0.33
NPC1 O15118 1/20 0.32
CASP3 P42574 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15445381 0.83 SGMS2 (0.31) ESR1SGMS2
SCHEMBL2610141 0.81 ALDH1A1 (0.43) TSHRALDH1A1LMNAMAPTSGMS2
SCHEMBL3295518 0.81 ALDH1A1 (0.36) ALDH1A1MEN1LMNAMAPTKMT2A
SCHEMBL30154222 0.81 IDO1 (0.34) ALDH1A1LMNACYP2C19
SCHEMBL11042257 0.81 ALDH1A1 (0.42) TSHRALDH1A1MAPTNPSR1SGMS2
SCHEMBL18501011 0.79 ESR1 (0.47) ESR1TSHRALDH1A1MEN1LMNA
SCHEMBL11041678 0.79 GAA (0.35) ALDH1A1MEN1KMT2AGAA
SCHEMBL9827673 0.79 ALDH1A1 (0.33) ALDH1A1LMNASGMS2
SCHEMBL7085423 0.78 ALDH1A1 (0.42) ALDH1A1MEN1MAPTKMT2AADRA2A
SCHEMBL11043231 0.78 AR (0.37) SLC6A4ACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101885742-B Chiral diphosphorodiamidate compound and synthesis method thereof UNIV HEFEI TECHNOLOGY 2013-01-09 CN disclosed
CN-101962391-B Chiral phosphorus compound UNIV HEFEI TECHNOLOGY 2012-09-26 CN disclosed
US-8163947-B2 Cyanation catalyst and method for producing optically active cyanhydrin compound using the same NATIONAL UNIVERSITY CORPORATION, HOKKAIDO UNIVERSITY (JP) 2012-04-24 US disclosed
CN-101973952-A Chiral oxazoline and synthetic method thereof UNIV HEFEI TECHNOLOGY 2011-02-16 CN disclosed
CN-101962391-A Chiral phosphorus compound UNIV HEFEI TECHNOLOGY 2011-02-02 CN disclosed
CN-101885742-A Chiral diphosphorodiamidate compound and synthesis method thereof UNIV HEFEI TECHNOLOGY 2010-11-17 CN disclosed
US-20100029977-A1 CYANATION CATALYST AND METHOD FOR PRODUCING OPTICALLY ACTIVE CYANHYDRIN COMPOUND USING THE SAME NATIONAL UNIVERSITY CORPORATION HOKKAIDO UNIVERSITY (JP) 2010-02-04 US disclosed
US-5449682-A Angiotensin II antagonists incorporating a substituted benzyl element MERCK & CO., INC. (US) 1995-09-12 US disclosed
US-5240938-A Angiotensin II antagonists incorporating a substituted pyridoimidazolyl ring MERCK & CO., INC. (US) 1993-08-31 US disclosed
WO-1991011999-A1 ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO., INC. (US) 1991-08-22 WO disclosed
US-4448971-A Hypoglycemic 5-phenyl-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1984-05-15 US disclosed
US-4407811-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1983-10-04 US disclosed
US-4399296-A TRIMETHYLSILYL CYANOHYDRIN INTERMEDIATES PFIZER INC. (US) 1983-08-16 US disclosed
US-4367234-A HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1983-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029977-A1 CYANATION CATALYST AND METHOD FOR PRODUCING OPTICALLY ACTIVE CYANHYDRIN COMPOUND USING THE SAME TYR, IK, CYB5R3 ESR1 2732/4885TSHR 1007/4885ALDH1A1 2995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.