SCHEMBL26106524

SCHEMBL26106524

Clc1nc(Cl)c2c(Br)nn(C3CCOCC3)c2n1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 6/20 0.35
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CG P48736 1/20 0.32
CSNK1A1 P48729 1/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32
CFTR P13569 1/20 0.32
RET P07949 2/20 0.31
PDE4D Q08499 1/20 0.31
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE1C Q14123 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30298010 1.00 NR3C1 (0.35) NR3C1PIK3CDPIK3CAPIK3CGCSNK1A1
SCHEMBL21631562 0.77 YTHDC1 (0.40) RET
SCHEMBL30297955 0.73 PLK4 (0.50)
SCHEMBL26505011 0.73 PLK4 (0.50)
SCHEMBL31194647 0.71 KDM4E (0.47) NR3C1CFTR
SCHEMBL15353927 0.71 CNR2 (0.37) PIK3CAPIK3CGPDE4DPDE1APDE1B
SCHEMBL173599 0.70 PDE1C (0.50) PDE4DPDE1APDE1BPDE1C
SCHEMBL31194579 0.69 KDM4E (0.55) NR3C1PIK3CDPIK3CAPIK3CGCFTR
SCHEMBL31194609 0.69 KDM4E (0.51) NR3C1PIK3CDPIK3CAPIK3CGCFTR
SCHEMBL31194551 0.68 ALDH1A1 (0.57) NR3C1CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116023380-B Pyrazolopyrimidine derivative, and preparation method and application thereof 沈阳药科大学 2024-01-23 CN disclosed
WO-2023071218-A1 PYRAZOLOPYRIMIDINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 沈阳药科大学 2023-05-04 WO disclosed
WO-2023071218-A1 PYRAZOLOPYRIMIDINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 沈阳药科大学 2023-05-04 WO disclosed
CN-116023380-A Pyrazolopyrimidine derivative, and preparation method and application thereof 沈阳药科大学 2023-04-28 CN disclosed